HA130 pentaacetate 70 and 200 nM for

70 and 200 nM for IKKβ

Smiles: CC1(C)C[C@H]2C3=CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@@]4(C)[C@]3(C)C[C@@H](O)[C@]2(CC1)C(O)=O

CAS Number: 2360527-40-6

Chemical Name: acetyl-L-leucyl-L-tryptophyl-L-tyrosyl-L-threonyl-L-aspartyl-L-isoleucyl-L-arginyl-L-methionyl-L-seryl-L-tryptophyl-L-arginyl-L-valyl-L-proline--acetic acid (1/1)

the elevation of intracellular calcium and the upregulation of NOS

HA130 pentaacetate 70 and 200 nM forHA130 is a selective autotaxin (ATX) inhibitor with an IC50 of 28 nM. Product information CAS Number: 1229652 21 4 Molecular Weight: 463. 29 Formula: C24H19BFNO5S Chemical Name: (3 {[4 ({3 [(4 fluorophenyl)methyl] 2, 4 dioxo 1, 3 thiazolidin 5 ylidene}methyl)phenoxy]methyl}phenyl)boronic acid Smiles: OB(O)C1=CC(COC2C=CC(C=C3SC(=O)N(CC4C=CC(F)=CC=4)C3=O)=CC=2)=CC=C1 InChiKey: VTNKMYWFWQTEHE XKZIYDEJSA N InChi: InChI=1S C24H19BFNO5S c26 20 8 4 17(5 9