Chemical Name: N-(3-chlorophenyl)-6
3 nM for PDGFRα
Naphthoquinone components from Alkanna tinctoria (L
injection of 15 mg MKT-077 1kg body weight each day for 5 days is significantly lower than that of untreated controls
SLC13A5-IN-1 exhibits an IC50 of 100 μM in recombinant Human GlyT2/3H-Glycine Uptake Assay
(R)-Elagolix Size:Contact [email protected] for quotation Chemical Name: N-(3-chlorophenyl)-6Elagolix is a highly potent, selective, orally active, short duration, non peptide antagonist of the gonadotropin releasing hormone receptor (GnRHR) (KD = 54 pM). Target: GnRHin vitro: Elagolix is a short acting, nonpeptide, GnRH antagonist, administered orally, that unlike injectable depot GnRH agonists and antagonists, produces a dose dependent suppression of ovarian estrogen production, that is, from partial suppression at lower doses to full